PROTAC BRD4 Degrader-5 Catalog No.:M8001-10 Mubritinib displays no inhibitory activities

Mubritinib displays no inhibitory activities against PC-3 cells with HER2 expressed very faintly with IC50 of 4

InChiKey: ZOPOQLDXFHBOIH-UHFFFAOYSA-N

using 32P-NAD+ as substrate

Molecular Weight: 599

fridge or bench shelf

PROTAC BRD4 Degrader-5 Catalog No.:M8001-10 Mubritinib displays no inhibitory activitiesPROTAC BRD4 Degrader 5 is a PROTAC based BRD4 degrader. PROTAC BRD4 Degrader 5 can potent degrade BRD4 in HER2 positive and negative breast cancer cell lines. Product information CAS Number: 2409538 70 9 Molecular Weight: 1016. 67 Formula: C50H62ClN9O8S2 Chemical Name: (2S, 4R) 1 [(2S) 2 (2 {2 [2 (2 {2 [(9S) 7 (4 chlorophenyl) 4, 5, 13 trimethyl 3 thia 1, 8, 11, 12 tetraazatricyclo[8. 3. 0. 0, ]trideca 2(6), 4, 7, 10, 12 pentaen 9